EPI-001

Name: EPI-001
SKU: A15814
Price: 175 CNY
Rating: 5 (288 reviews)

目录号: A15814

Androgen Receptor 拮抗剂

EPI-001 是一种雄激素受体（AR）的拮抗剂，通过与 AR 的 N-末端结构域（NTD）共价结合并阻断 AR 及其剪接变体的转录活性所需的蛋白-蛋白相互作用（抑制 AR NTD 转录激活的 IC50 约为 6 微摩尔）。

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Grouped product items
规格	价格	库存
2mg	¥175.00	现货
5mg	¥245.00	现货
10mg	¥455.00	现货
25mg	¥840.00	现货
50mg	¥1,435.00	现货
100mg	¥2,170.00	现货
200mg	¥3,255.00	现货
*10mM 1mL in DMSO**	¥280.00	现货
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Data Sheet

SDS

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生物活性

Discription

EPI-001 is an antagonist of the androgen receptor (AR) that acts by binding covalently to the N-terminal domain (NTD) of the AR and blocking protein-protein interactions required for transcriptional activity of the AR and its splice variants (IC50 for inhibition of AR NTD transactivation ?? 6 μM)

Targets

Target	Value

产品信息

目录号	A15814
分子式	C21H27ClO5
分子量	394.89
CAS号	227947-06-0
SMILES	CC(C)(C1=CC=C(C=C1)OCC(CO)O)C2=CC=C(C=C2)OCC(CCl)O
其他名称	EPI001, EPI 001
储存条件	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

溶解性数据

In vitro	DMSO	72 mg/mL (182.32 mM)
	Water	Insoluble
	Ethanol	72 mg/mL (182.32 mM)
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	25.32 mL	126.62 mL	253.24 mL
0.5 mM	5.06 mL	25.32 mL	50.65 mL
1 mM	2.53 mL	12.66 mL	25.32 mL
5 mM	0.51 mL	2.53 mL	5.06 mL

Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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* Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C₁V₁ = C₂V₂

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