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￥ 0.00 Pim
| Catalog No. | Inhibitor Name | Pim1 | Pim2 | Pim3 | Other |
|---|---|---|---|---|---|
| A10838 | SGI-1776 free base | *** | * | * | FLT3 |
| A11945 | SMI-4a | ** | |||
| A14275 | CX-6258 HCl | *** | ** | ** | |
| A13203 | AZD1208 | **** | *** | **** | |
| A11967 | TCS PIM-1 4a | ** | * | ||
| A12896 | CX-6258 | *** | ** | ** | |
| A15368 | PIM-1 Inhibitor 2 | * | |||
| A15369 | TCS PIM-1 1 | * |
Notes:
1.Hover mouse over "" to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of "" is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.
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SGI-1776 (free base)
Catalog No. A10838 PIM1 抑制剂SGI-1776 (free base)是Pim1的一种新型ATP竞争性抑制剂，在无细胞试验中的IC50为7 nM，选择性是Pim2和Pim3的50倍和10倍，对Flt3和haspin也有效。阶段1。 了解更多
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