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Ertiprotafib

Ertiprotafib

Name: Ertiprotafib
SKU: A20815

目录号: A20815

PTP1B/IKK-βinhibitor and dual PPARα and PPARβ agonist

Ertiprotafib Chemical Structure

CAS NO. 251303-04-5

Ertiprotafib is an inhibitor of PTP1B, IkB kinase β (IKK-β), and a dual PPARα and PPARβ agonist, with an IC50 of 1.6 μM for PTP1B, 400 nM for IKK-β, an EC50 of ~1 μM for PPARα/PPARβ.

库存：现货

规格	价格	数量
1 mg	￥ 3,200.00
5 mg	￥ 9,600.00
10 mg	￥ 16,000.00

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产品仅用于科学研究，不针对患者销售，望谅解.

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生物活性

Ertiprotafib is an inhibitor of PTP1B, IkB kinase β (IKK-β), and a dual PPARα and PPARβ agonist, with an IC50 of 1.6 μM for PTP1B, 400 nM for IKK-β, an EC50 of ~1 μM for PPARα/PPARβ.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	17.87 mL	89.36 mL	178.73 mL
0.5 mM	3.57 mL	17.87 mL	35.75 mL
1 mM	1.79 mL	8.94 mL	17.87 mL
5 mM	0.36 mL	1.79 mL	3.57 mL

*The above data is based on the productmolecular weight 559.51. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A20815
M. Wt	559.51
Formula	C31H27BrO3S
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	251303-04-5
Synonyms	PTP 112, PTP112, PTP-112
SMILES	OC([C@@H](CC1=CC=CC=C1)OC2=C(C)C=C(C3=C(C(C)=C(C)S4)C4=C(Br)C5=CC=CC=C53)C=C2C)=O