ESI-09
目录号: A14233
EPAC1/EPAC2 抑制剂
ESI-09 是一种特异性的直接由 cAMP 激活的交换蛋白(EPAC)抑制剂,对 EPAC1 和 EPAC2 的 IC50 分别为 3.2 uM 和 1.4 uM。
Discription | ESI-09 is a specific exchange protein directly activated by cAMP (EPAC) inhibitor with IC50 of 3.2 uM and 1.4 uM for EPAC1 and EPAC2, | |||||
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Targets |
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Cell Research |
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目录号 | A14233 |
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分子式 | C16H15ClN4O2 |
分子量 | 330.77 |
CAS号 | 263707-16-0 |
SMILES | CC(C)(C)C1=CC(=NO1)C(=O)/C(=N/NC2=CC(=CC=C2)Cl)/C#N |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro (25°C) | DMSO | 63 mg/mL (190.46 mM) | |
Water | Insoluble | ||
Ethanol | Warmed: 19 mg/mL (57.44 mM) | ||
In vivo | 10% ethanol+10% Tween 80+ddH2O | 1 mg/mL | |
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 30.23 mL | 151.16 mL | 302.32 mL |
0.5 mM | 6.05 mL | 30.23 mL | 60.46 mL |
1 mM | 3.02 mL | 15.12 mL | 30.23 mL |
5 mM | 0.6 mL | 3.02 mL | 6.05 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2