Fedovapagon
目录号: A21286
V2R 激动剂
Fedovapagon 是一种选择性的加压素 V2 受体(V2R)激动剂,其 EC50 为 24 nM,目前正在开发中,用于治疗夜尿症。
| Discription | Fedovapagon is a selective vasopressin V2 receptor (V2R) agonist with an EC50 of 24 nM, which is being developed for the treatment of nocturia. | |||||
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| 目录号 | A21286 |
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| 分子式 | C27H34N4O3 |
| 分子量 | 462.58 |
| CAS号 | 347887-36-9 |
| SMILES | CC1=C(CNC(N2CCC[C@]2(C(N(C)C)=O)[H])=O)C=CC(C(N3CCCCC4=C3C=CC=C4)=O)=C1 |
| 储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2