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G Protein

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AMG 837

Catalog No. A21160
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GPR40 agonist

AMG 837 is a potent GPR40 agonist(EC50=13 nM) with a superior pharmacokinetic profile and robust glucose-dependent stimulation of insulin secretion in rodents. 了解更多

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MK-0354

Catalog No. A22008
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GPR109a receptor agonist

MK-0354 is a partial agonist of GPR109a receptor, for hGPR109a/ mGPR109a with EC50 of 1.65/1.08 μM, showed no activation of GPR109b. 了解更多

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AMG 837 sodium salt

Catalog No. A21793
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GPR40 agonist

AMG 837 sodium salt is a potent GPR40 agonist(EC50=13 nM) with a superior pharmacokinetic profile and robust glucose-dependent stimulation of insulin secretion in rodents. 了解更多

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AM-4668

Catalog No. A21778
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GPR40 agonist

AM-4668 is a GPR40 agonist for type 2 diabetes. EC50s of 3.6 nM and 36 nM for GPR40 in A9 cells (GPR40 IP3 assay) and CHO cells (GPR40 aequorin assay), respectively. 了解更多

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(1R,2R)-2-PCCA(hydrochloride)

Catalog No. A21655
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GPR88 receptor agonist

(1R,2R)-2-PCCA hydrochloride is a diastereomer of 2-PCCA, and acts as a potent GPR88 receptor agonist, with an EC50 of 3 nM in cell-free assay, and 603 nM in cell assay. 了解更多

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AF64394

Catalog No. A21574
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GPR3 inverse agonist

AF64394 is a GPR3 inverse agonist, with a pIC50 of 7.3. 了解更多

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AM-1638

Catalog No. A21505
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GPR40/FFA1 full agonist

AM-1638 is a potent and orally bioavailable GPR40/FFA1 full agonist with an EC50 of 0.16 μM. 了解更多

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PSN632408

Catalog No. A20902
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GPR119 receptors agonist

PSN632408 is an optimized agonist of GPR119 receptors that shows similar potency to OEA at both recombinant mouse and human GPR119 receptors, exhibiting EC50 values of 5.6 and 7.9 uM, respectively. 了解更多

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Kynurenic acid sodium

Catalog No. A20000
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GPR35/CXCR8 agonist

Kynurenic acid sodium, an endogenous tryptophan metabolite, is a broad-spectrum antagonist targeting NMDA, glutamate, α7 nicotinic acetylcholine receptor. Kynurenic acid sodium is also an agonist of GPR35/CXCR8. 了解更多

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GPR35 agonist 1

Catalog No. A12462
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GPR35/CXCR8 agonist

GPR35 agonist 1 (compound 50) is a potent and specific G protein-coupled receptor-35 (GPR35)/CXCR8 agonist with an EC50 of 5.8 nM, displays good druggability. 了解更多

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LY2922470

Catalog No. A12181
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GPR40 agonist

LY2922470 is a potent, selective and orally available agonist of the G protein-coupled receptor 40 (GPR40), with EC50s of 7 nM, 1 nM and 3 nM for human GPR40, mouse GPR40 and rat GPR40, respectively. 了解更多

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DJ-V-159

Catalog No. A18853
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GPRC6A agonist

DJ-V-159 is an agonist for G protein-coupled receptor family C group 6 member A (GPRC6A). 了解更多

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Kynurenic acid

Catalog No. A16581
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GPR35/CXCR8 拮抗剂

Kynurenic acid, an endogenous tryptophan metabolite, is a broad-spectrum antagonist targeting NMDA, glutamate, α7 nicotinic acetylcholine receptor. Kynurenic acid is also an agonist of GPR35/CXCR8. 了解更多

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TM N1324

Catalog No. A17038
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GPR39 激动剂

TM N1324是G蛋白偶联受体39（GPR39）的激动剂，在Zn2+存在下的EC50为9 nM/5 nM，而对于人/鼠GPR39，则在Zn2+不存在时的EC50为280 nM/180 nM。了解更多

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MK-6892

Catalog No. A12982
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GPR109A 激动剂

MK-6892是高亲和力烟酸（NA）受体GPR109A的有效，选择性和完全激动剂。人GPR109A的MK-6892的Ki和GTPγSEC 50分别为4 nM和16 nM。了解更多

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