GABA Receptors

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Gabazine

Catalog No. A12627
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GABAA receptor antagonist

Gabazine is a selective and competitive antagonist of GABAA receptor, with an IC50 of ~0.2 μM for GABA receptor. 了解更多

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SCH 50911

Catalog No. A21630
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γ-Aminobutyric acid B GABA(B) receptor antagonist

SCH 50911, (+)-(S)-5,5-dimethylmorpholinyl-2-acetic acid, a selective, orally-active and competitive γ-Aminobutyric acid B GABA(B) receptor antagonist. 了解更多

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U-93631

Catalog No. A16336
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GABAA receptor ligand

U-93631是具有新颖化学结构的GABAA受体配体，IC50为100 nM，并且已显示在重组GABAA受体中诱导GABA诱导的全细胞Cl-电流快速，时间依赖性地衰减。了解更多

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(-)-Securinine

Catalog No. A17102
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GABA receptor 拮抗剂

(-)-Securinine是一种最初从S. suffructicosa分离的生物碱。Securinine是一种特定的GABA受体拮抗剂，已发现在体内具有显着的CNS活性。了解更多

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Cgp 52432

Catalog No. A17140
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GABA-A receptor 拮抗剂

Cgp 52432是GABA-A受体拮抗剂。了解更多

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CGP 36742

Catalog No. A18666
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GABAB receptor antagonist

CGP 36742 is a selective GABAB receptor antagonist that can penetrate the blood?Cbrain barrier after peripheral administration, with an IC50 of 32?μM. CGP 36742 is useful in treatment of depression. 了解更多

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Flumazenil

Catalog No. A10397
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Benzodiazepine 拮抗剂

Flumazenil是竞争性抑制GABA/苯二氮卓受体复合物上苯二氮卓识别位点的活性。Flumazenil在一些活性动物模型中是弱部分激动剂，但在人类中很少或没有激动剂活性。了解更多

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(+)-Bicuculline

Catalog No. A12590
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GABAA 拮抗剂

(+)-Bicuculline是一种经典的GABAA拮抗剂。了解更多

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- Maryam Adenike Salaudeen, .et al. Anticonvulsant Activity of Tapinanthus dodoneifolius (DC.) Danser in Chicks and Mice: A Potential Source of Novel Anticonvulsant Agent, J Pharmacy and Drug Innovations, 2022, 3(4)
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2-Hydroxysaclofen

Catalog No. A13696
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GABAB receptors 拮抗剂

2-Hydroxysaclofen对GABAB受体是一种有效的选择性拮抗剂。了解更多

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Cloflubicyne

Catalog No. A13932
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GABA 拮抗剂

Cloflubicyne是一种有效的非竞争性GABA拮抗剂，惊厥药，实验室杀虫剂。了解更多

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RO 15-3890

Catalog No. A14349
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benzodiazepine receptor 拮抗剂

Ro 15-1788是苯二氮卓受体拮抗剂。了解更多

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Picrotoxin

Catalog No. A14004
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GABAA receptor 拮抗剂

Picrotoxin是GABAA受体拮抗剂。该化合物已显示可增加下丘脑的去甲肾上腺素水平和周转率。了解更多

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- Maryam Adenike Salaudeen, .et al. Anticonvulsant Activity of Tapinanthus dodoneifolius (DC.) Danser in Chicks and Mice: A Potential Source of Novel Anticonvulsant Agent, J Pharmacy and Drug Innovations, 2022, 3(4)