GKT137831

目录号: A14433

NOX1/4 inhibitor

GKT137831 Chemical Structure

CAS NO. 1218942-37-0

GKT137831 is a first in class inhibitor targeting NOX1 and NOX4 enzymes.

库存: 现货

规格 价格 数量
5 mg
¥ 900.00
10 mg
¥ 1,400.00
25 mg
¥ 3,200.00
10mM * 1mL in DMSO
¥ 1,000.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

详情

GKT137831 is a first in class inhibitor targeting NOX1 and NOX4 enzymes.
Targets
NOX1 NOX4
110 nM(Ki)140 nM(Ki)
In vitro DMSO 78 mg/mL heating (197.54 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 25.33 mL 126.63 mL 253.26 mL
0.5 mM 5.07 mL 25.33 mL 50.65 mL
1 mM 2.53 mL 12.66 mL 25.33 mL
5 mM 0.51 mL 2.53 mL 5.07 mL

*The above data is based on the productmolecular weight 394.85. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A14433
MECHANISM OF ACTION Inhibitor
M. Wt 394.85
Formula C21H19ClN4O2
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1218942-37-0
Synonyms GKT-137831, GKT 137831
SMILES CN1C(=O)C=C2C(=C1C3=CC(=CC=C3)N(C)C)C(=O)N(N2)C4=CC=CC=C4Cl

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