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GKT137831

促销

NOX1/4 抑制剂

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产品目录号: A14433

库存状态:中国现货中国现货

产品名 目录号 价格 数量
GKT137831 5mg A14433-5
¥ 900.00
GKT137831 10mg A14433-10
¥ 1,400.00
GKT137831 25mg A14433-25
¥ 3,200.00
GKT137831 10mM * 1mL in DMSO A14433-10mM-D
¥ 1,000.00

产品仅用于研究,不针对患者销售,望谅解.

产品简介

GKT137831 is a first in class inhibitor targeting NOX1 and NOX4 enzymes.

GKT137831

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Chemical Information

目录号 A14433
Mechanism of action Inhibitor
分子量 394.85
化学分子式 C21H19ClN4O2
Solubility DMSO
纯度 >98%
储存方式 at -20°C 2 years
CAS No. 1218942-37-0
Synonyms GKT-137831, GKT 137831
SMILES code CN1C(=O)C=C2C(=C1C3=CC(=CC=C3)N(C)C)C(=O)N(N2)C4=CC=CC=C4Cl
化学名称 N/A

生物活性

Description
GKT137831 is a first in class inhibitor targeting NOX1 and NOX4 enzymes.
Targets
NOX1 NOX4
110 nM(Ki)140 nM(Ki)

溶解性

Solubility (25°C)* In vitro DMSO 78 mg/mL heating (197.54 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 25.33 mL 126.63 mL 253.26mL
0.5 mM 5.07 mL 25.33 mL 50.65 mL
1 mM 2.53 mL 12.66 mL 25.33 mL
5 mM 0.51 mL 2.53 mL 5.07 mL

*The above data is based on the productmolecular weight 394.85. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

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