Glycyl-H 1152 2HCl
目录号: A13659
ROCK 抑制剂
Glycyl-H 1152 2HCl 是一种选择性且高效的 ROCK 抑制剂(IC50 值分别为 0.0118、2.35、2.57、3.26、>10 和 >10 uM,针对 ROCKII、Aurora A、CAMKII、PKG、PKA 和 PKC)。
Discription | Glycyl-H 1152 2HCl is a selective and potent ROCK inhibitor (IC50 values are 0.0118, 2.35, 2.57, 3.26, > 10 and >10 uM for ROCKII, Aurora A, CAMKII, PKG, PKA and PKC respectively.) | ||
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Targets |
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目录号 | A13659 |
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分子式 | C18H24N4O3S.2HCl |
分子量 | 449.4 |
CAS号 | 913844-45-8 |
SMILES | C[C@H]1CN(CCCN1S(=O)(=O)C2=CC=CC3=C2C(=CN=C3)C)C(=O)CN.Cl.Cl |
其他名称 | Rho Kinase Inhibitor IV |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2