GNE-207

目录号: A18844

CBP bromodomain inhibitor

GNE-207

GNE-207 Chemical Structure

CAS NO. 2158266-58-9

GNE-207 is a novel, potent, and orally bioavailable inhibitor of the bromodomain of CBP. GNE-207 has excellent CBP potency (CBP IC50?=?1?nM, MYC EC50?=?18?nM), and it exhibits a good pharmacokinetic profile.

库存: 现货

规格 价格 数量
1 mg
¥ 5,000.00
5 mg
¥ 9,200.00
10 mg
¥ 13,800.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

产品详情

GNE-207 is a novel, potent, and orally bioavailable inhibitor of the bromodomain of CBP. GNE-207 has excellent CBP potency (CBP IC50?=?1?nM, MYC EC50?=?18?nM), and it exhibits a good pharmacokinetic profile.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 19.58 mL 97.92 mL 195.85 mL
0.5 mM 3.92 mL 19.58 mL 39.17 mL
1 mM 1.96 mL 9.79 mL 19.58 mL
5 mM 0.39 mL 1.96 mL 3.92 mL

*The above data is based on the productmolecular weight 510.6. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A18844
作用机制 Inhibitor (抑制剂)
M. Wt 510.6
Formula C29H30N6O3
Purity >99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No. 2158266-58-9
Synonyms GNE207, GNE 207
SMILES O=C(NC)C1=NC=C(C2=CC3=C(C=N2)C(C4=NN(C5CCOCC5)C6=C4CN(C(C)=O)CC6)=CC=C3)C=C1

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