CCG258208 hydrochloride (GRK2-IN-1)

Name: CCG258208 hydrochloride (GRK2-IN-1)
SKU: A20131
Price: 2205 CNY
Rating: 5 (288 reviews)

目录号: A20131

GRKs-IN-1，化合物14as，对G蛋白偶联受体激酶2 GRK2（IC50=30 nM）和GRK5（IC50=7.1 μM）具有显著的效力和选择性。GRKs-IN-1是帕罗西汀的衍生物14as，在心肌细胞收缩性测试中比帕罗西汀提高了100倍。

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Grouped product items
规格	价格	库存
1mg	¥2,205.00	现货
5mg	¥2,520.00	现货
10mg	¥3,990.00	现货
25mg	¥7,245.00	现货
50mg	¥12,075.00	现货
100mg	¥16,485.00	现货
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Data Sheet

SDS

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生物活性

Discription

GRKs-IN-1, Compound 14as, has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50=30 nM) and GRK5 (IC50=7.1 μM). GRKs-IN-1 is a derivative 14as of paroxetine, shows a 100-fold improvement in cardiomyocyte contractility assays over paroxetine.

Targets

Target	Value

产品信息

目录号	A20131
分子式	C24H25FN4O4
分子量	452.48
CAS号	2055990-90-2
SMILES	FC1=C(C(NCC2=NNC=C2)=O)C=C([C@H]3[C@H](COC4=CC=C(OCO5)C5=C4)CNCC3)C=C1
储存条件	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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