GS967
目录号: A14361
late INa 抑制剂
GS967 是一种新型、高效、选择性的心脏晚期钠电流（晚期 INa）抑制剂；在心室肌细胞和分离心脏中抑制 ATX-II 引起的晚期 I(Na)，其 IC(50) 值分别为 0.13 和 0.21 微摩尔。
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生物活性
| Discription | GS967 is a novel, potent, and selective inhibitor of cardiac late sodium current(late INa); inhibits ATX-II-induced late I(Na) in ventricular myocytes and isolated hearts with IC(50) values of 0.13 and 0.21 uM, respectively. | |||||
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| Cell Research |
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产品信息
| 目录号 | A14361 |
|---|---|
| 分子式 | C14H7F6N3O |
| 分子量 | 347.22 |
| CAS号 | 1262618-39-2 |
| SMILES | FC(F)(F)C1=NN=C2C=CC(C3=CC=C(OC(F)(F)F)C=C3)=CN21 |
| 其他名称 | GS-967, GS 967 |
| 储存条件 | Store lyophilized at -20ºC, keep desiccated. |
溶解性数据
| In vitro | DMSO | 38 mg/mL (109.44 mM) | |
| Water | Insoluble | ||
| Ethanol | 39 mg/mL (112.32 mM) | ||
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* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
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Preparing Stock Solutions
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 28.8 mL | 144 mL | 288 mL |
| 0.5 mM | 5.76 mL | 28.8 mL | 57.6 mL |
| 1 mM | 2.88 mL | 14.4 mL | 28.8 mL |
| 5 mM | 0.58 mL | 2.88 mL | 5.76 mL |
Useful Calculator
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2
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| 购买 1262618-39-2 | 1262618-39-2 供应商 | 1262618-39-2 花费 | 1262618-39-2 生产商 | 订购 1262618-39-2 | 1262618-39-2 代理商