GSK 4027
目录号: A12531
GSK 4027 是 PCAF/GCN5 溴结构域的化学探针,在时间分辨荧光共振能量转移(TR-FRET)测定中,对 PCAF 的 pIC50 为 7.4±0.11。
| Discription | GSK 4027 is a chemical probe for the PCAF/GCN5 bromodomain with an pIC50 of 7.4??0.11 for PCAF in a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. | |||||
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| Cell Research |
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| 目录号 | A12531 |
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| 分子式 | C17H21BrN4O |
| 分子量 | 377.28 |
| CAS号 | 2079896-25-4 |
| SMILES | BrC1=C(N[C@@H]2C[C@H](C3=CC=CC=C3)CN(C)C2)C=NN(C)C1=O |
| 其他名称 | GSK4027, GSK-4027 |
| 储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2