GSK1059615

目录号: A10438

mTOR/PI3K 抑制剂

GSK1059615

GSK1059615 Chemical Structure

CAS NO. 958852-01-2

GSK1059615是PI3Kα (IC50 = 2 nM)的强效、可逆、ATP竞争性噻唑烷二酮抑制剂。

库存: 现货

规格 价格 数量
5 mg
¥ 700.00
10 mg
¥ 1,200.00
25 mg
¥ 2,500.00
50 mg
¥ 4,500.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

产品详情

GSK1059615是PI3Kα (IC50 = 2 nM)的强效、可逆、ATP竞争性噻唑烷二酮抑制剂。
靶点信息
PI3Kα PI3Kβ PI3Kδ PI3Kγ mTOR
0.4 nM0.6 nM2 nM5 nM12 nM
In vitro DMSO 2 mg/mL (5.99 mM)
Water Insoluble
Ethanol Insoluble
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 29.99 mL 149.97 mL 299.94 mL
0.5 mM 6 mL 29.99 mL 59.99 mL
1 mM 3 mL 15 mL 29.99 mL
5 mM 0.6 mL 3 mL 6 mL

*The above data is based on the productmolecular weight 333.4 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A10438
作用机制 Inhibitor (抑制剂)
M. Wt 333.4
Formula C18H11N3O2S
Purity >99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No. 958852-01-2
Synonyms GSK-1059615
SMILES C1=CC2=NC=CC(=C2C=C1/C=C\3/C(=O)NC(=O)S3)C4=CC=NC=C4

产品标签

产品标签

其他人对该产品使用了下列标签:

使用空格分隔标签。使用单引号(')标注词组。

Product Questions

Product Questions

No Questions
Keywords:购买 GSK1059615 | GSK1059615 供应商 | 订购 GSK1059615 | GSK1059615 价格 | GSK1059615 生产商 | 订单 GSK1059615 | GSK1059615 代理商 | 购买 958852-01-2| 958852-01-2 供应商 | 订购 958852-01-2 | 958852-01-2 价格 | 958852-01-2 生产商 | 订单 958852-01-2 | 958852-01-2 代理商|buy GSK1059615 | GSK1059615 Supplier | purchase GSK1059615 | GSK1059615 cost | GSK1059615 manufacturer | order GSK1059615 | GSK1059615 distributor | buy 958852-01-2| 958852-01-2 Supplier | purchase 958852-01-2 | 958852-01-2 cost | 958852-01-2 manufacturer | order 958852-01-2 | 958852-01-2 distributor
Rewards