GSK126

目录号: A11757

EZH2 抑制剂

GSK126

GSK126 Chemical Structure

CAS NO. 1346574-57-9

GSK126是一种有效的,高选择性的,具有S-腺苷甲硫氨酸竞争性的小分子EZH2甲基转移酶活性抑制剂,可降低总体H3K27me3水平并重新激活沉默的PRC2目标基因。

库存: 现货

规格 价格 数量
2 mg
¥ 400.00
5 mg
¥ 600.00
10 mg
¥ 900.00
25 mg
¥ 1,600.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

产品详情

GSK126是一种有效的,高选择性的,具有S-腺苷甲硫氨酸竞争性的小分子EZH2甲基转移酶活性抑制剂,可降低总体H3K27me3水平并重新激活沉默的PRC2目标基因。
靶点信息
EZH2
9.9 nM
In vitro (25°C) DMSO Warmed: 3 mg/mL (5.69 mM)
Water Insoluble
Ethanol Insoluble
In vivo 4% DMSO+corn oil 0.4 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 18.99 mL 94.94 mL 189.87 mL
0.5 mM 3.8 mL 18.99 mL 37.97 mL
1 mM 1.9 mL 9.49 mL 18.99 mL
5 mM 0.38 mL 1.9 mL 3.8 mL

*The above data is based on the productmolecular weight 526.67. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A11757
作用机制 Inhibitor (抑制剂)
M. Wt 526.67
Formula C31H38N6O2
Purity >99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No. 1346574-57-9
Synonyms GSK 126, GSK-126
SMILES CC[C@H](C)N1C=C(C2=C(C=C(C=C21)C3=CN=C(C=C3)N4CCNCC4)C(=O)NCC5=C(C=C(NC5=O)C)C)C

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