GSK1324726A (I-BET726)

目录号: A14133

BET 抑制剂

GSK1324726A (I-BET726)

GSK1324726A (I-BET726) Chemical Structure

CAS NO. 1300031-52-0

GSK1324726A (I-BET726)是一种新型、高效、选择性的BET蛋白小分子抑制剂,对BRD2(IC50 = 41 nM)、BRD3(IC50 = 31 nM)和BRD4(IC50 = 22 nM)具有高度的亲和力。

库存: 现货

规格 价格 数量
5 mg
¥ 1,040.00
10 mg
¥ 1,770.00
25 mg
¥ 3,120.00
10mM * 1mL in DMSO
¥ 1,650.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

产品详情

GSK1324726A (I-BET726)是一种新型、高效、选择性的BET蛋白小分子抑制剂,对BRD2(IC50 = 41 nM)、BRD3(IC50 = 31 nM)和BRD4(IC50 = 22 nM)具有高度的亲和力。
靶点信息
BRD4 BRD3 BRD2
22 nM31 nM41 nM
In vitro DMSO 77 mg/mL (177.05 mM)
Water Insoluble
Ethanol 77 mg/mL (177.05 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 22.99 mL 114.97 mL 229.93 mL
0.5 mM 4.6 mL 22.99 mL 45.99 mL
1 mM 2.3 mL 11.5 mL 22.99 mL
5 mM 0.46 mL 2.3 mL 4.6 mL

*The above data is based on the productmolecular weight 434.91. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A14133
作用机制 Inhibitor (抑制剂)
M. Wt 434.91
Formula C25H23ClN2O3
Purity >99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No. 1300031-52-0
Synonyms I-BET726, GSK 1324726A, GSK-1324726A, I-BET 726
SMILES CC1CC(C2=C(N1C(=O)C)C=CC(=C2)C3=CC=C(C=C3)C(=O)O)NC4=CC=C(C=C4)Cl

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