GSK2126458 (Omipalisib)

Name: GSK2126458 (Omipalisib)
SKU: A11035
Price: 245 CNY
Rating: 5 (288 reviews)

目录号: A11035

mTOR/PI3K 抑制剂,

GSK2126458 是一种高效、口服生物利用度的 PI3Kα 和 mTOR 抑制剂，在体内药效动力学和肿瘤生长效能模型中均显示活性。

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Grouped product items
规格	价格	库存
2mg	¥245.00	现货
5mg	¥385.00	现货
10mg	¥630.00	现货
25mg	¥1,225.00	现货
50mg	¥1,960.00	现货
100mg	¥2,940.00	现货
*10mM 1mL in DMSO**	¥385.00	现货
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Data Sheet

SDS

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生物活性

Discription

GSK2126458 is a highly potent, orally bioavailable inhibitor of PI3Kα and mTOR with in vivo activity in both pharmacodynamic and tumor growth efficacy models.

Targets

Target	Value

Cell Research

Cell Line	Type	Value	Description	References

产品信息

目录号	A11035
分子式	C25H17F2N5O3S
分子量	505.5
CAS号	1086062-66-9
SMILES	COC1=C(C=C(C=N1)C2=CC3=C(C=CN=C3C=C2)C4=CN=NC=C4)NS(=O)(=O)C5=C(C=C(C=C5)F)F
其他名称	GSK-2126458
储存条件	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

溶解性数据

In vitro (25°C)	DMSO	96 mg/mL (189.91 mM)
	Water	Insoluble
	Ethanol	Insoluble
In vivo	2% DMSO+40% PEG 300+2% Tween 80+ddH2O	3 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	19.78 mL	98.91 mL	197.82 mL
0.5 mM	3.96 mL	19.78 mL	39.56 mL
1 mM	1.98 mL	9.89 mL	19.78 mL
5 mM	0.4 mL	1.98 mL	3.96 mL

Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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* Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C₁V₁ = C₂V₂

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