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GSK221149A (Retosiban)

GSK221149A (Retosiban)

Name: GSK221149A (Retosiban)
SKU: A13106

目录号: A13106

Oxytocin Receptor 拮抗剂

GSK221149A (Retosiban) Chemical Structure

CAS NO. 820957-38-8

GSK221149A (Retosiban)是一种口服药物，可作为选择性纳摩尔（Ki = 0.65 nM）催产素受体拮抗剂，其选择性是相关血管加压素受体的> 1400倍。

库存：缺货

规格	价格
5 mg	￥ 3,500.00
10 mg	￥ 6,000.00
25 mg	￥ 12,000.00
50 mg	￥ 20,000.00

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产品仅用于科学研究，不针对患者销售，望谅解.

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生物活性

GSK221149A (Retosiban)是一种口服药物，可作为选择性纳摩尔（Ki = 0.65 nM）催产素受体拮抗剂，其选择性是相关血管加压素受体的> 1400倍。

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	20.22 mL	101.1 mL	202.19 mL
0.5 mM	4.04 mL	20.22 mL	40.44 mL
1 mM	2.02 mL	10.11 mL	20.22 mL
5 mM	0.4 mL	2.02 mL	4.04 mL

*The above data is based on the productmolecular weight 494.58. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A13106
作用机制	Antagonist (拮抗剂)
M. Wt	494.58
Formula	C27H34N4O5
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	820957-38-8
Synonyms	GSK-221149A, GSK 221149A
SMILES	CC[C@H](C)[C@@H]1C(=O)N[C@@H](C(=O)N1[C@H](C2=COC(=N2)C)C(=O)N3CCOCC3)C4CC5=CC=CC=C5C4