Trusted by 10,000+ Scientists since 2006
微信关注
申请试用装

GSK256066 2,2,2-trifluoroacetic acid

PDE 抑制剂

0 Customer Reviews
产品目录号: A15097

库存状态:中国现货中国现货

产品名 目录号 价格 数量
GSK256066 2,2,2-trifluoroacetic acid 10mg A15097-10
¥ 2,000.00
GSK256066 2,2,2-trifluoroacetic acid 50mg A15097-50
¥ 6,000.00
GSK256066 2,2,2-trifluoroacetic acid 500mg A15097-500
¥ 17,000.00

产品仅用于研究,不针对患者销售,望谅解.

产品简介

GSK256066 is a selective PDE4B(equal affinity to isoforms A-D) inhibitor with IC50 of 3.2 pM, >380,000-fold selectivity versus PDE1/2/3/5/6 and >2500-fold selectivity against PDE4B versus PDE7.

GSK256066 2,2,2-trifluoroacetic acid

双击上述图片即可查看完整大小

缩小
放大

更多视图

顾客使用 Adooq 产品发表的高质量科研文献

Chemical Information

目录号 A15097
Mechanism of action Inhibitor
分子量 632.61
化学分子式 C29H27F3N4O7S
Solubility DMSO
纯度 >98%
储存方式 at -20°C 2 years
CAS No. 1415560-64-3
Synonyms GSK-256066, GSK 256066
SMILES code CC1=C2C(=CC(=C1)S(=O)(=O)C3=CC=CC(=C3)C(=O)N(C)C)C(=C(C=N2)C(=O)N)NC4=CC(=CC=C4)OC.C(=O)(C(F)(F)F)O
化学名称 6-[3-(dimethylcarbamoyl)phenyl]sulfonyl-4-(3-methoxyanilino)-8-methylquinoline-3-carboxamide;2,2,2-trifluoroacetic acid

生物活性

Description
GSK256066 is a selective PDE4B(equal affinity to isoforms A-D) inhibitor with IC50 of 3.2 pM, >380,000-fold selectivity versus PDE1/2/3/5/6 and >2500-fold selectivity against PDE4B versus PDE7.

制备储备液

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 15.81 mL 79.04 mL 158.08mL
0.5 mM 3.16 mL 15.81 mL 31.62 mL
1 mM 1.58 mL 7.9 mL 15.81 mL
5 mM 0.32 mL 1.58 mL 3.16 mL

*The above data is based on the productmolecular weight 632.61. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Ordering online

To place an order online, simply browse to the product you are interested in and click on the 'Add to Cart' button. To complete this process, you will need to confirm the size and quantity of the products that you require.

To complete an order you will need to register using our simple online registration process. We do not share your contact details with any third parties.

When you are ready to check out simply enter your PO number to complete the ordering process. Please ensure that you send us a copy of your PO by fax or email afterwards.  We will then liaise with you or your purchasing department to confirm the order.

Found your products but not ready to order?

Why not use our WishList feature to store lists of products? This convenient feature allows you to manage lists, append notes to products and share lists with co-workers or colleagues.

Ordering offline

You can email or fax us your purchase order and we will place the order for you. You can also phone us to place the order.  Our contact details are:

We require the following information to process your order:
  • The catalog number for each product. 
  • Your email address or fax number. 
  • Your name and telephone number. 
  • Shipping address and billing address.
  • Purchase order numbers.

产品标签

使用空格分隔标签。使用单引号(')标注词组。


Keywords:购买 GSK256066 2,2,2-trifluoroacetic acid | GSK256066 2,2,2-trifluoroacetic acid 供应商 | 订购 GSK256066 2,2,2-trifluoroacetic acid | GSK256066 2,2,2-trifluoroacetic acid 价格 | GSK256066 2,2,2-trifluoroacetic acid 生产商 | 订单 GSK256066 2,2,2-trifluoroacetic acid | GSK256066 2,2,2-trifluoroacetic acid 代理商 | 购买 1415560-64-3| 1415560-64-3 供应商 | 订购 1415560-64-3 | 1415560-64-3 价格 | 1415560-64-3 生产商 | 订单 1415560-64-3 | 1415560-64-3 代理商|buy GSK256066 2,2,2-trifluoroacetic acid | GSK256066 2,2,2-trifluoroacetic acid Supplier | purchase GSK256066 2,2,2-trifluoroacetic acid | GSK256066 2,2,2-trifluoroacetic acid cost | GSK256066 2,2,2-trifluoroacetic acid manufacturer | order GSK256066 2,2,2-trifluoroacetic acid | GSK256066 2,2,2-trifluoroacetic acid distributor | buy 1415560-64-3| 1415560-64-3 Supplier | purchase 1415560-64-3 | 1415560-64-3 cost | 1415560-64-3 manufacturer | order 1415560-64-3 | 1415560-64-3 distributor