GSK256066

目录号: A11073

PDE Inhibitor

GSK256066

GSK256066 Chemical Structure

CAS NO. 801312-28-7

GSK256066 is an exceptionally high affinity and selective inhibitor of PDE4 that inhibits PDE4 isoforms A-D with equal affinity and has a high HARBS (High-Affinity Rolipram Binding Site) ratio (>17).

库存: 现货

规格 价格 数量
5 mg
¥ 1,200.00
10 mg
¥ 2,200.00
50 mg
¥ 6,000.00
100 mg
¥ 9,800.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

详情

GSK256066 is an exceptionally high affinity and selective inhibitor of PDE4 that inhibits PDE4 isoforms A-D with equal affinity and has a high HARBS (High-Affinity Rolipram Binding Site) ratio (>17).
Targets
PDE4B
3.2 pM
In vitro (25°C) DMSO 5 mg/mL (9.64 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 30% propylene glycol, 5% Tween 80, 65% D5W 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 19.28 mL 96.41 mL 192.83 mL
0.5 mM 3.86 mL 19.28 mL 38.57 mL
1 mM 1.93 mL 9.64 mL 19.28 mL
5 mM 0.39 mL 1.93 mL 3.86 mL

*The above data is based on the productmolecular weight 518.6. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Technical Details

目录号 A11073
MECHANISM OF ACTION Inhibitor
M. Wt 518.6
Formula C27H26N4O5S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 801312-28-7
Synonyms GSK-256066
SMILES CC1=C2C(=CC(=C1)S(=O)(=O)C3=CC=CC(=C3)C(=O)N(C)C)C(=C(C=N2)C(=O)N)NC4=CC(=CC=C4)OC

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