GSK2606414

目录号: A12792

PERK 抑制剂

GSK2606414 Chemical Structure

CAS NO. 1337531-36-8

GSK2606414是口服有效的选择性PERK抑制剂,IC50为0.4 nM。

库存: 现货

规格 价格 数量
5 mg
¥ 850.00
10 mg
¥ 1,150.00
25 mg
¥ 2,250.00
50 mg
¥ 3,350.00
10mM * 1mL in DMSO
¥ 1,490.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

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GSK2606414是口服有效的选择性PERK抑制剂,IC50为0.4 nM。
靶点信息
EIF2AK3 (PERK) (Cell-free assay) EIF2AK1 (HRI) (Cell-free assay) EIF2AK2 (PKR) (Cell-free assay)
0.4 nM420 nM696 nM
In vitro DMSO 90 mg/mL (199.36 mM)
Water <1 mg/mL (<1 mM)
Ethanol 19 mg/mL (42.08 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 22.15 mL 110.76 mL 221.51 mL
0.5 mM 4.43 mL 22.15 mL 44.3 mL
1 mM 2.22 mL 11.08 mL 22.15 mL
5 mM 0.44 mL 2.22 mL 4.43 mL

*The above data is based on the productmolecular weight 451.44. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A12792
MECHANISM OF ACTION Inhibitor
M. Wt 451.44
Formula C24H20F3N5O
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1337531-36-8
Synonyms GSK-2606414, GSK 2606414
SMILES CN1C=C(C2=C1N=CN=C2N)C3=CC4=C(C=C3)N(CC4)C(=O)CC5=CC(=CC=C5)C(F)(F)F

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