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PERK 抑制剂

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产品目录号: A12792


产品名 目录号 价格 数量
GSK2606414 5mg A12792-5
¥ 850.00
GSK2606414 10mg A12792-10
¥ 1,150.00
GSK2606414 25mg A12792-25
¥ 2,250.00
GSK2606414 50mg A12792-50
¥ 3,350.00
GSK2606414 10mM * 1mL in DMSO A12792-10mM-D
¥ 1,490.00



GSK2606414 is an orally available, potent, and selective PERK inhibitor with IC50 of 0.4 nM.





顾客使用 Adooq 产品发表的高质量科研文献

Chemical Information

目录号 A12792
Mechanism of action Inhibitor
分子量 451.44
化学分子式 C24H20F3N5O
Solubility DMSO
纯度 >98%
储存方式 at -20°C 2 years
CAS No. 1337531-36-8
Synonyms GSK-2606414, GSK 2606414
SMILES code CN1C=C(C2=C1N=CN=C2N)C3=CC4=C(C=C3)N(CC4)C(=O)CC5=CC(=CC=C5)C(F)(F)F
化学名称 7Methyl-5-(1-{[3-(trifluoroMethyl)phenyl]acetyl}-2,3-dihydro1Hindol-5-yl)7Hpyrrolo[2,3d]pyriMidin-4-aMine


GSK2606414 is an orally available, potent, and selective PERK inhibitor with IC50 of 0.4 nM.
EIF2AK3 (PERK) (Cell-free assay) EIF2AK1 (HRI) (Cell-free assay) EIF2AK2 (PKR) (Cell-free assay)
0.4 nM420 nM696 nM


Solubility (25°C)* In vitro DMSO 90 mg/mL (199.36 mM)
Water <1 mg/mL (<1 mM)
Ethanol 19 mg/mL (42.08 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.


Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 22.15 mL 110.76 mL 221.51mL
0.5 mM 4.43 mL 22.15 mL 44.3 mL
1 mM 2.22 mL 11.08 mL 22.15 mL
5 mM 0.44 mL 2.22 mL 4.43 mL

*The above data is based on the productmolecular weight 451.44. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

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