GSK2656157

Name: GSK2656157
SKU: A13577
Price: 175 CNY
Rating: 5 (3 reviews)

目录号: A13577

PERK 抑制剂

3 篇发表文献

GSK2656157 是一种与 ATP 竞争的 PERK 酶活性抑制剂，其 IC(50) 为 0.9 nmol/L。它对 PERK 具有高度选择性，其 IC(50) 值在针对 300 种激酶的测试中均 >100 nmol/L。

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Grouped product items
规格	价格	库存
2mg	¥175.00	现货
5mg	¥315.00	现货
10mg	¥455.00	现货
25mg	¥980.00	现货
50mg	¥1,715.00	现货
100mg	¥2,765.00	现货
200mg	¥4,620.00	现货
*10mM 1mL in DMSO**	¥490.00	现货
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重要通知：仅供研究使用。我们不向患者销售。

Data Sheet

SDS

顾客使用 Adooq 产品发表的高质量科研文献

Adooq用户使用GSK2656157发表的3篇文献

Jun Liu, .et al. , Food Chem, 2023, Jun 30;412:135550 PMID: 36706507

Cao W, .et al. , J Cell Mol Med, 2019, Aug 23 PMID: 31441588

Kosuke Ishikawa, .et al. , Biology Methods and Protocols, 2018, 1-10

生物活性

Discription

GSK2656157 is an ATP-competitive inhibitor of PERK enzyme activity with an IC(50) of 0.9 nmol/L. It is highly selective for PERK with IC(50) values >100 nmol/L against a panel of 300 kinases.

Targets

Target	Value

Cell Research

Cell Line	Type	Value	Description	References

产品信息

目录号	A13577
分子式	C23H21FN6O
分子量	416.45
CAS号	1337532-29-2
SMILES	CC1=NC(=CC=C1)CC(=O)N2CCC3=C2C=CC(=C3F)C4=CN(C5=C4C(=NC=N5)N)C
其他名称	GSK 2656157
储存条件	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

溶解性数据

In vitro (25°C)	DMSO	28 mg/mL (67.23 mM)
	Water	Insoluble
	Ethanol	Insoluble
In vivo	1% CMC Na	28 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	24.01 mL	120.06 mL	240.12 mL
0.5 mM	4.8 mL	24.01 mL	48.02 mL
1 mM	2.4 mL	12.01 mL	24.01 mL
5 mM	0.48 mL	2.4 mL	4.8 mL

Useful Calculator

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Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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* Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C₁V₁ = C₂V₂

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