GSK461364

目录号: A10442

PLK Inhibitor

GSK461364

GSK461364 Chemical Structure

CAS NO. 929095-18-1

GSK461364 is an ATP-competitive inhibitor of polo-like kinase 1 (Plk1).

库存: 现货

规格 价格 数量
5 mg
¥ 800.00
10 mg
¥ 1,500.00
25 mg
¥ 3,000.00
50 mg
¥ 4,800.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

详情

GSK461364 is an ATP-competitive inhibitor of polo-like kinase 1 (Plk1).
Targets
PLK1 (Cell-free assay)
2.2 nM(Ki)
In vitro (25°C) DMSO 10 mg/mL (18.39 mM)
Water <1 mg/mL (<1 mM)
Ethanol 30 mg/mL (55.18 mM)
In vivo 1% DMSO/30% polyethylene glycol/1% Tween 80 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 18.4 mL 91.98 mL 183.96 mL
0.5 mM 3.68 mL 18.4 mL 36.79 mL
1 mM 1.84 mL 9.2 mL 18.4 mL
5 mM 0.37 mL 1.84 mL 3.68 mL

*The above data is based on the productmolecular weight 543.6 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Technical Details

目录号 A10442
MECHANISM OF ACTION Inhibitor
M. Wt 543.6
Formula C27H28F3N5O2S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 929095-18-1
Synonyms GSK 461364, GSK-461364
SMILES C[C@H](C1=CC=CC=C1C(F)(F)F)OC2=C(SC(=C2)N3C=NC4=C3C=C(C=C4)CN5CCN(CC5)C)C(=O)N

产品标签

产品标签

其他人对该产品使用了下列标签:

使用空格分隔标签。使用单引号(')标注词组。

Product Questions

Product Questions

No Questions
Keywords:购买 GSK461364 | GSK461364 供应商 | 订购 GSK461364 | GSK461364 价格 | GSK461364 生产商 | 订单 GSK461364 | GSK461364 代理商 | 购买 929095-18-1| 929095-18-1 供应商 | 订购 929095-18-1 | 929095-18-1 价格 | 929095-18-1 生产商 | 订单 929095-18-1 | 929095-18-1 代理商|buy GSK461364 | GSK461364 Supplier | purchase GSK461364 | GSK461364 cost | GSK461364 manufacturer | order GSK461364 | GSK461364 distributor | buy 929095-18-1| 929095-18-1 Supplier | purchase 929095-18-1 | 929095-18-1 cost | 929095-18-1 manufacturer | order 929095-18-1 | 929095-18-1 distributor
Rewards