GSK467

Name: GSK467
SKU: A18807
Price: 385 CNY
Rating: 5 (288 reviews)

目录号: A18807

KDM5B (JARID1B or PLU1) 抑制剂

GSK467 是一种强效且选择性的 KDM5（也称为 JARID1）抑制剂，其 Ki 值为 10 nM，对 KDM4C 的选择性高达 180 倍，并且对 KDM6 或其他 Jumonji 家族成员没有可测量的抑制效果。GSK467 利用独特的结合模式。

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Grouped product items
规格	价格	库存
1mg	¥385.00	现货
5mg	¥1,015.00	现货
10mg	¥1,540.00	现货
25mg	¥2,940.00	现货
50mg	¥4,585.00	现货
100mg	¥6,195.00	现货
*10mM 1mL in DMSO**	¥1,330.00	现货
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Data Sheet

SDS

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生物活性

Discription

GSK467 is a potent and selective inhibitor of KDM5 (also known as JARID1) with a Ki of 10 nM, shows 180-fold selectivity for KDM4C and no measurable inhibitory effects toward KDM6 or other Jumonji family members. GSK467 exploits unique binding modes.

Targets

Target	Value

Cell Research

Cell Line	Type	Value	Description	References

产品信息

目录号	A18807
分子式	C17H13N5O2
分子量	319.32
CAS号	1628332-52-4
SMILES	O=C1C2=C(C=NC=C2)N=C(OC3=CN(CC4=CC=CC=C4)N=C3)N1
其他名称	GSK467; GSK-467; GSK 467;
储存条件	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

溶解性数据

In vitro	DMSO	7 mg/mL (21.92 mM)
	Water	<1 mg/mL
	Ethanol	<1 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	31.32 mL	156.58 mL	313.17 mL
0.5 mM	6.26 mL	31.32 mL	62.63 mL
1 mM	3.13 mL	15.66 mL	31.32 mL
5 mM	0.63 mL	3.13 mL	6.26 mL

Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

Calculate Reset

* Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C₁V₁ = C₂V₂

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