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GSK5182

GSK5182

Name: GSK5182
SKU: A19383

目录号: A19383

ERRγ agonist

Product Citations (1)

GSK5182 Chemical Structure

CAS NO. 877387-37-6

GSK5182 is a highly selective inverse agonist of estrogen-related receptor γ (ERRγ) with an IC50 of 79 nM and does not interact with other nuclear receptors, including ERRα or ERα.

库存：现货

规格	价格	数量
1 mg	￥ 800.00
5 mg	￥ 2,500.00
10 mg	￥ 4,100.00

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生物活性

GSK5182 is a highly selective inverse agonist of estrogen-related receptor γ (ERRγ) with an IC50 of 79 nM and does not interact with other nuclear receptors, including ERRα or ERα.

溶解度 *

In vitro	DMSO	78 mg/mL
	Water	Insoluble
	Ethanol	78 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	23.95 mL	119.75 mL	239.5 mL
0.5 mM	4.79 mL	23.95 mL	47.9 mL
1 mM	2.39 mL	11.97 mL	23.95 mL
5 mM	0.48 mL	2.39 mL	4.79 mL

*The above data is based on the productmolecular weight 417.54. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A19383
作用机制	Agonist (激动剂)
M. Wt	417.54
Formula	C27H31NO3
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	877387-37-6
Synonyms	GSK 5182, GSK-5182
SMILES	OCCC/C(C1=CC=CC=C1)=C(C2=CC=C(O)C=C2)/C3=CC=C(OCCN(C)C)C=C3