GSK690693

目录号: A11030

AKT 抑制剂

GSK690693

GSK690693 Chemical Structure

CAS NO. 937174-76-0

GSK690693是一种新型的ATP竞争性低纳摩尔泛Akt激酶抑制剂(IC50值分别为Akt1、2和3的2、13和9 nM)。

库存: 现货

规格 价格 数量
10 mg
¥ 1,200.00
25 mg
¥ 2,200.00
50 mg
¥ 3,600.00
100 mg
¥ 6,000.00
10mM * 1mL in DMSO
¥ 750.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

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GSK690693是一种新型的ATP竞争性低纳摩尔泛Akt激酶抑制剂(IC50值分别为Akt1、2和3的2、13和9 nM)。
Targets
Target Value
Akt1IC50: 2nM
PKCηIC50: 2nM
PKCθIC50: 2nM
PrkXIC50: 5nM
Akt3IC50: 9nM
Akt2IC50: 13nM
PKCδIC50: 14nM
PKCβIC50: 19nM
PKCεIC50: 21nM
PKAIC50: 24nM
PKG1βIC50: 33nM
In vitro (25°C) DMSO 36 mg/mL (84.61 mM)
Water Insoluble
Ethanol Insoluble
In vivo 5% DMSO+40%PEG300+5% tween80+50% H2O 2 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 23.5 mL 117.51 mL 235.02 mL
0.5 mM 4.7 mL 23.5 mL 47 mL
1 mM 2.35 mL 11.75 mL 23.5 mL
5 mM 0.47 mL 2.35 mL 4.7 mL

*The above data is based on the productmolecular weight 425.5 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A11030
作用机制 Inhibitor (抑制剂)
M. Wt 425.5
Formula C21H27N7O3
Purity >99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No. 937174-76-0
Synonyms GSK-690693
SMILES CCN1C2=C(C(=NC=C2OC[C@H]3CCCNC3)C#CC(C)(C)O)N=C1C4=NON=C4N

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