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GW842166X

CB2 receptor 激动剂

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产品目录号: A11253

库存状态:中国现货中国现货

产品名 目录号 价格 数量
GW842166X 5mg A11253-5
¥ 600.00
GW842166X 10mg A11253-10
¥ 1,000.00
GW842166X 25mg A11253-25
¥ 2,000.00
GW842166X 10mM * 1mL in DMSO A11253-10mM-D
¥ 1,130.00

产品仅用于研究,不针对患者销售,望谅解.

产品简介

GW842166X is a selective non-cannabinoid CB2 receptor agonist, which is undergoing clinical development as a novel oral treatment for inflammatory pain

GW842166X

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Chemical Information

目录号 A11253
Mechanism of action Agonist
分子量 449.25
化学分子式 C18H17Cl2F3N4O2
Solubility DMSO
纯度 >98%
储存方式 at -20°C 2 years
CAS No. 666260-75-9, 956013-38-0
Synonyms N/A
SMILES code C1COCCC1CNC(=O)C2=CN=C(N=C2C(F)(F)F)NC3=C(C=C(C=C3)Cl)Cl
化学名称 2-(2,4-dichlorophenylamino)-N-((tetrahydro-2H-pyran-4-yl)methyl)-4-(trifluoromethyl)pyrimidine-5-carboxamide

生物活性

Description
GW842166X is a selective non-cannabinoid CB2 receptor agonist, which is undergoing clinical development as a novel oral treatment for inflammatory pain
Targets
CB2
63 nM(EC50)

溶解性

Solubility (25°C) * In vitro DMSO 20 mg/mL (44.51 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 30% propylene glycol, 5% Tween 80, 65% D5W 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 22.26 mL 111.3 mL 222.59mL
0.5 mM 4.45 mL 22.26 mL 44.52 mL
1 mM 2.23 mL 11.13 mL 22.26 mL
5 mM 0.45 mL 2.23 mL 4.45 mL

*The above data is based on the productmolecular weight 449.25. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

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