微信关注
Total item
Cart Subtotal
￥ 0.00 产品详情
GW 9508是一种可透过细胞的氨基苯基丙酸酯，可作为G蛋白偶联受体（GPCR）GRP40/FFA1受体（EC50?50 nM）的有效选择性激动剂，对家族成员GRP120的活性降低（EC50?3.5μM），GRP41/GRP43（EC50> 50μM），以及一组八种其他游离脂肪酸（FFA）和前列腺素受体。
靶点信息
| GPR40 | GPR120 | |||
| 7.32(pEC50) | 5.46(pEC50) |
| In vitro (25°C) | DMSO | 63 mg/mL (181.34 mM) | |
| Water | Insoluble | ||
| Ethanol | 63 mg/mL (181.34 mM) | ||
| In vivo | 2% DMSO+40% PEG 300+2% Tween 80+ddH2O | 1 mg/mL | |
|
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
|||
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 28.79 mL | 143.93 mL | 287.85 mL |
| 0.5 mM | 5.76 mL | 28.79 mL | 57.57 mL |
| 1 mM | 2.88 mL | 14.39 mL | 28.79 mL |
| 5 mM | 0.58 mL | 2.88 mL | 5.76 mL |
*The above data is based on the productmolecular weight 347.4. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| 目录号 | A11965 |
|---|---|
| 作用机制 | Inhibitor (抑制剂) |
| M. Wt | 347.4 |
| Formula | C22H21NO3 |
| Purity | >99% |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
| CAS No. | 885101-89-3 |
| Synonyms | GW 9508, GW-9508 |
| SMILES | C1=CC=C(C=C1)OC2=CC=CC(=C2)CNC3=CC=C(C=C3)CCC(=O)O |
产品标签
Product Questions
Product Questions
No Questions
Keywords:购买 GW9508 | GW9508 供应商 | 订购 GW9508 | GW9508 价格 | GW9508 生产商 | 订单 GW9508 | GW9508 代理商 | 购买 885101-89-3| 885101-89-3 供应商 | 订购 885101-89-3 | 885101-89-3 价格 | 885101-89-3 生产商 | 订单 885101-89-3 | 885101-89-3 代理商|buy GW9508 | GW9508 Supplier | purchase GW9508 | GW9508 cost | GW9508 manufacturer | order GW9508 | GW9508 distributor | buy 885101-89-3| 885101-89-3 Supplier | purchase 885101-89-3 | 885101-89-3 cost | 885101-89-3 manufacturer | order 885101-89-3 | 885101-89-3 distributor