INK 128 (MLN0128)

目录号: A11461

mTOR inhibitor

INK 128 (MLN0128)

INK 128 (MLN0128) Chemical Structure

CAS NO. 1224844-38-5

INK 128 is a TORC1/2 inhibitor, is also an orally bioavailable inhibitor of raptor-mTOR (TOR complex 1 or TORC1) and rictor-mTOR (TOR complex 2 or TORC2) with potential antineoplastic activity.

库存: 现货

规格 价格 数量
5 mg
¥ 800.00
10 mg
¥ 1,000.00
25 mg
¥ 1,800.00
50 mg
¥ 2,500.00
10mM * 1mL in DMSO
¥ 800.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

详情

INK 128 is a TORC1/2 inhibitor, is also an orally bioavailable inhibitor of raptor-mTOR (TOR complex 1 or TORC1) and rictor-mTOR (TOR complex 2 or TORC2) with potential antineoplastic activity.
Targets
Target Value
mTORki: 1.4nM
mTORki: 1.4nM
PI3KαIC50: 219nM
PI3KγIC50: 221nM
PI3KδIC50: 230nM
PI3KβIC50: 5293nM
In vitro (25°C) DMSO 62 mg/mL (200.43 mM)
Water <1 mg/mL (<1 mM)
Ethanol 2 mg/mL (6.46 mM)
In vivo 30% PEG400/0.5% Tween80/5% propylene glycol 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 32.33 mL 161.66 mL 323.31 mL
0.5 mM 6.47 mL 32.33 mL 64.66 mL
1 mM 3.23 mL 16.17 mL 32.33 mL
5 mM 0.65 mL 3.23 mL 6.47 mL

*The above data is based on the productmolecular weight 309.3 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A11461
MECHANISM OF ACTION Inhibitor
M. Wt 309.3
Formula C15H15N7O
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1224844-38-5
Synonyms INK128, INK-128
SMILES CC(C)N1C2=C(C(=N1)C3=CC4=C(C=C3)OC(=N4)N)C(=NC=N2)N

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