Ipragliflozin
目录号: A13556
SGLT2 抑制剂
Ipragliflozin 是一种高效且选择性的 SGLT2 抑制剂,其 IC50 为 2.8 nM;对 SGLT1/3/4/5/6 几乎没有抑制作用。
| Discription | Ipragliflozin is a highly potent and selective SGLT2 inhibitor with IC50 of 2.8 nM; little and NO potency for SGLT1/3/4/5/6. | |||||
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| Cell Research |
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| 目录号 | A13556 |
|---|---|
| 分子式 | C21H21FO5S |
| 分子量 | 404.4559 |
| CAS号 | 761423-87-4 |
| SMILES | C1=CC=C2C(=C1)C=C(S2)CC3=C(C=CC(=C3)[C@H]4[C@@H]([C@H]([C@@H]([C@H](O4)CO)O)O)O)F |
| 其他名称 | ASP 1941, ASP1941 |
| 储存条件 | Store lyophilized at -20ºC, keep desiccated. |
| In vitro | DMSO | 78 mg/mL (192.85 mM) | |
| Water | Insoluble | ||
| Ethanol | 78 mg/mL (192.85 mM) | ||
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* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
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| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 24.72 mL | 123.62 mL | 247.25 mL |
| 0.5 mM | 4.94 mL | 24.72 mL | 49.45 mL |
| 1 mM | 2.47 mL | 12.36 mL | 24.72 mL |
| 5 mM | 0.49 mL | 2.47 mL | 4.94 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2