JAK3-IN-1
目录号: A20734
JAK3 抑制剂
JAK3-IN-1 是一种强效的 JAK3 抑制剂,其 IC50 为 4.8 nM,同时也能抑制 JAK1(IC50 = 896 nM)和 JAK2(IC50 = 1050 nM)。
Discription | JAK3-IN-1 is a potent JAK3 inhibitor with IC50 of 4.8 nM, also inhibits JAK1 (IC50 = 896 nM) and JAK2 (IC50 = 1050 nM). | |||||
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Targets |
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Cell Research |
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目录号 | A20734 |
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分子式 | C26H30ClN7O2 |
分子量 | 508.02 |
CAS号 | 1805787-93-2 |
SMILES | O=C(C=C)NC1=CC(CNC2=NC(NC3=C(OC)C=C(N4CCN(C)CC4)C=C3)=NC=C2Cl)=CC=C1 |
其他名称 | JAK3IN1; JAK3 IN 1; JAK3IN-1; JAK3-IN1 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2