JD-5037
目录号: A20837
CB1R 拮抗剂
JD-5037 是一种新型的周围限制性 CB1R 拮抗剂,其 IC50 为 1.5 nM。
| Discription | JD-5037 is a novel, peripherally restricted CB1R antagonist with an IC50 of 1.5 nM. | ||
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| Targets |
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| 目录号 | A20837 |
|---|---|
| 分子式 | C27H27Cl2N5O3S |
| 分子量 | 572.51 |
| CAS号 | 1392116-14-1 |
| SMILES | NC([C@H](C(C)C)/N=C(NS(=O)(C1=CC=C(Cl)C=C1)=O)\N2N=C(C3=CC=C(Cl)C=C3)[C@@H](C4=CC=CC=C4)C2)=O |
| 其他名称 | JD5037, JD 5037 |
| 储存条件 | Store lyophilized at -20ºC, keep desiccated. |
| In vitro | DMSO | 90 mg/mL (157.19 mM) | |
| Water | Insoluble | ||
| Ethanol | 2 mg/mL (3.49 mM) | ||
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* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
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| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 17.47 mL | 87.33 mL | 174.67 mL |
| 0.5 mM | 3.49 mL | 17.47 mL | 34.93 mL |
| 1 mM | 1.75 mL | 8.73 mL | 17.47 mL |
| 5 mM | 0.35 mL | 1.75 mL | 3.49 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2