JNJ16259685
目录号: A20545
mGlu1 receptor 拮抗剂
JNJ16259685 是一种选择性的 mGlu1 受体 拮抗剂,能够以浓度依赖的方式抑制 mGlu1 的突触激活,其 IC50 为 19 nM。
Discription | JNJ16259685 is a selective antagonist of mGlu1 receptor, and inhibits the synaptic activation of mGlu1 in a concentration-dependent manner with IC50 of 19 nM. | ||
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目录号 | A20545 |
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分子式 | C20H23NO3 |
分子量 | 325.4 |
CAS号 | 409345-29-5 |
SMILES | O=C(C1=CC=C2N=C3C(CCCO3)=CC2=C1)[C@H]4CC[C@@H](OC)CC4 |
其他名称 | JNJ 16259685; JNJ-16259685 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2