Kenpaullone

目录号: A11220

CDK inhibitor

Kenpaullone

Kenpaullone Chemical Structure

CAS NO. 142273-20-9

Kenpaullone is a potent inhibitor of CDK1/cyclin B (IC₅₀ = 400 nM), CDK2/cyclin A (IC₅₀ = 680nM) , CDK5 (IC₅₀ = 850nM) and with much less effect other kinases.

库存: 现货 Shipped in 7-10 Days

规格 价格 数量
10 mg
¥ 900.00
50 mg
¥ 3,800.00
100 mg
¥ 6,500.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

详情

Kenpaullone is a potent inhibitor of CDK1/cyclin B (IC₅₀ = 400 nM), CDK2/cyclin A (IC₅₀ = 680nM) , CDK5 (IC₅₀ = 850nM) and with much less effect other kinases.
Targets
Target Value
GSK-3βIC50: 0.23μM
CDK1/CyclinBIC50: 0.4μM
CDK2/CyclinAIC50: 0.68μM
CDK5/p35IC50: 0.85μM
CDK2/CyclinEIC50: 7.5μM
ERK2IC50: 9μM
c-SrcIC50: 15μM
CaseinKinase2IC50: 20μM
ERK1IC50: 20μM
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 30.56 mL 152.81 mL 305.62 mL
0.5 mM 6.11 mL 30.56 mL 61.12 mL
1 mM 3.06 mL 15.28 mL 30.56 mL
5 mM 0.61 mL 3.06 mL 6.11 mL

*The above data is based on the productmolecular weight 327.2. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A11220
MECHANISM OF ACTION Inhibitor
M. Wt 327.2
Formula C16H11BrN2O
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 142273-20-9
Synonyms N/A
SMILES C1C2=C(C3=CC=CC=C3NC1=O)NC4=C2C=C(C=C4)Br

产品标签

产品标签

使用空格分隔标签。使用单引号(')标注词组。

Product Questions

Product Questions

No Questions
您还可能对下列产品感兴趣
Keywords:购买 Kenpaullone | Kenpaullone 供应商 | 订购 Kenpaullone | Kenpaullone 价格 | Kenpaullone 生产商 | 订单 Kenpaullone | Kenpaullone 代理商 | 购买 142273-20-9| 142273-20-9 供应商 | 订购 142273-20-9 | 142273-20-9 价格 | 142273-20-9 生产商 | 订单 142273-20-9 | 142273-20-9 代理商|buy Kenpaullone | Kenpaullone Supplier | purchase Kenpaullone | Kenpaullone cost | Kenpaullone manufacturer | order Kenpaullone | Kenpaullone distributor | buy 142273-20-9| 142273-20-9 Supplier | purchase 142273-20-9 | 142273-20-9 cost | 142273-20-9 manufacturer | order 142273-20-9 | 142273-20-9 distributor
Rewards