L-Moses (L-45)
目录号: A20587
BRD 抑制剂
L-45 是首个具有高效、选择性和细胞活性的 p300/CBP-associated factor (PCAF) bromodomain (Brd) 抑制剂,其 Kd 值为 126±15 nM。
Discription | L-45 is the first potent, selective, and cell-active p300/CBP-associated factor (PCAF) bromodomain (Brd) inhibitor with a Kd of 126±15 nM. | ||
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目录号 | A20587 |
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分子式 | C21H24N6 |
分子量 | 360.46 |
CAS号 | 2079885-05-3 |
SMILES | C[C@@H]([C@H](C1=CC=CC=C1)N(C)C)NC(C2=C3C=CC=C2)=NN4C3=NN=C4C |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2