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Lerociclib dihydrochloride

目录号: A21577
CDK4/CDK6 抑制剂
Lerociclib 二盐酸盐(G1T38 二盐酸盐)是一种强效且选择性的 CDK4/CDK6 抑制剂,其对 CDK4/CyclinD1CDK6/CyclinD3 的 IC50 分别为 1 nM 和 2 nM。
Grouped product items
规格 价格 库存 数量
1mg
¥175.00
现货
2mg
¥245.00
现货
5mg
¥455.00
现货
10mg
¥805.00
现货
50mg
¥3,255.00
现货
100mg
¥5,460.00
现货
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生物活性
Discription Lerociclib dihydrochloride (G1T38 dihydrochloride) is a potent and selective inhibitor of CDK4/CDK6, with IC50s of 1 nM and 2 nM for CDK4/CyclinD1 and CDK6/CyclinD3, respectively.
Targets
Target Value
产品信息
目录号 A21577
分子式 C26H36Cl2N8O
分子量 547.52
CAS号 2097938-59-3
SMILES O=C1NCC2(N3C1=CC4=CN=C(NC5=NC=C(N6CCN(C(C)C)CC6)C=C5)N=C43)CCCCC2.[H]Cl.[H]Cl
其他名称 G1T38 dihydrochloride, G1T 38, G1T-38
储存条件

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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    Volume

    Molecular Weight

Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C1V1 = C2V2

  • C1

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    C2

    V2

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