Lerociclib dihydrochloride
目录号: A21577
CDK4/CDK6 抑制剂
Lerociclib 二盐酸盐(G1T38 二盐酸盐)是一种强效且选择性的 CDK4/CDK6 抑制剂,其对 CDK4/CyclinD1 和 CDK6/CyclinD3 的 IC50 分别为 1 nM 和 2 nM。
Discription | Lerociclib dihydrochloride (G1T38 dihydrochloride) is a potent and selective inhibitor of CDK4/CDK6, with IC50s of 1 nM and 2 nM for CDK4/CyclinD1 and CDK6/CyclinD3, respectively. | ||
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目录号 | A21577 |
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分子式 | C26H36Cl2N8O |
分子量 | 547.52 |
CAS号 | 2097938-59-3 |
SMILES | O=C1NCC2(N3C1=CC4=CN=C(NC5=NC=C(N6CCN(C(C)C)CC6)C=C5)N=C43)CCCCC2.[H]Cl.[H]Cl |
其他名称 | G1T38 dihydrochloride, G1T 38, G1T-38 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2