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Lomitapide mesylate

Lomitapide mesylate

Name: Lomitapide mesylate
SKU: A16600

目录号: A16600

MTP inhibitor

Lomitapide mesylate Chemical Structure

CAS NO. 202914-84-9

Lomitapide mesylate(AEGR-733; BMS-201038) is an inhibitor of microsomal triglyceride-transfer protein (MTP) wtih in vitro IC50 of 8 nM.

库存：现货

规格	价格	数量
1 mg	￥ 3,200.00
5 mg	￥ 9,600.00
10 mg	￥ 16,000.00

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生物活性

Lomitapide mesylate(AEGR-733; BMS-201038) is an inhibitor of microsomal triglyceride-transfer protein (MTP) wtih in vitro IC50 of 8 nM.

溶解度 *

In vitro	DMSO	91 mg/mL (115.21 mM)
	Water	Insoluble
	Ethanol	91 mg/mL (115.21 mM)
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	12.66 mL	63.3 mL	126.61 mL
0.5 mM	2.53 mL	12.66 mL	25.32 mL
1 mM	1.27 mL	6.33 mL	12.66 mL
5 mM	0.25 mL	1.27 mL	2.53 mL

*The above data is based on the productmolecular weight 789.83. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A16600
作用机制	Inhibitor (抑制剂)
M. Wt	789.83
Formula	C40H41F6N3O5S
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	202914-84-9
Synonyms	AEGR-733 mesylate, AEGR733, AEGR 733; BMS-201038 mesylate, BMS 201038, BMS201038
SMILES	O=C(C1(CCCCN2CCC(NC(C3=CC=CC=C3C4=CC=C(C(F)(F)F)C=C4)=O)CC2)C5=C(C6=C1C=CC=C6)C=CC=C5)NCC(F)(F)F.O=S(C)(O)=O