LP-211
目录号: A16898
5-HT7 receptor 激动剂
LP-211 是一种选择性的 5-HT7 血清素受体激动剂,其在大鼠克隆的 5-HT7 受体上的 Ki 值为 0.58 nM,并且对 5-HT1A 受体的选择性超过 300 倍。
Discription | LP-211 is a a selective agonist of the serotonin 5-HT7 receptor with a Ki value of 0.58 nM at rat cloned 5-HT7 receptors, and >300-fold selectivity over the 5-HT1A receptor. | ||
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目录号 | A16898 |
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分子式 | C30H34N4O |
分子量 | 466.63 |
CAS号 | 1052147-86-0 |
SMILES | O=C(NCC1=CC=C(C#N)C=C1)CCCCCN2CCN(C3=CC=CC=C3C4=CC=CC=C4)CC2 |
其他名称 | LP211, LP 211 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2