LSD1-IN-6
目录号: A20474
LSD1 抑制剂
LSD1-IN-6(化合物4m)是一种强效且可逆的赖氨酸特异性去甲基化酶1(LSD1)抑制剂,其IC50为123 nM。LSD1-IN-6能增加组蛋白H3的二甲基赖氨酸4的水平,对LSD1的表达没有影响。
Discription | LSD1-IN-6 (Compound 4m) is a potent and reversible inhibitor of lysine-specific demethylase 1 (LSD1), with an IC50 of 123 nM. LSD1-IN-6 increases dimethylated Lys4 of histone H3, shows no effect on expression of LSD1. |
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目录号 | A20474 |
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分子式 | C15H13BrN2O3 |
分子量 | 349.18 |
CAS号 | 2035912-43-5 |
SMILES | OC1=C(O)C=C(Br)C(/C=C/C2=CC=C(/C(N)=N/O)C=C2)=C1 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2