Lurasidone (SM13496)

Name: Lurasidone (SM13496)
SKU: A11214

目录号: A11214

Dopamine D2 抑制剂

Lurasidone (SM13496) Chemical Structure

CAS NO. 367514-87-2

Lurasidone (SM-13496)是dopamine D2和5-HT7的拮抗剂，IC50 值分别为 1.68 和 0.495 nM。Lurasidone (SM-13496) 也是 5-HT1A 受体的部分激动剂。

库存：现货

规格	价格	数量
50 mg	￥ 900.00
100 mg	￥ 1,600.00
200 mg	￥ 3,000.00

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生物活性

Lurasidone (SM-13496)是dopamine D2和5-HT7的拮抗剂，IC50 值分别为 1.68 和 0.495 nM。Lurasidone (SM-13496) 也是 5-HT1A 受体的部分激动剂。

溶解度 *

In vitro	DMSO	7 mg/mL (14.2 mM)
	Water	Insoluble
	Ethanol	Insoluble
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	20.3 mL	101.48 mL	202.96 mL
0.5 mM	4.06 mL	20.3 mL	40.59 mL
1 mM	2.03 mL	10.15 mL	20.3 mL
5 mM	0.41 mL	2.03 mL	4.06 mL

*The above data is based on the productmolecular weight 492.7 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A11214
作用机制	Inhibitor (抑制剂)
M. Wt	492.7
Formula	C28H36N4O2S
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	367514-87-2
Synonyms	SM13496, SM-13496, SM 13496
SMILES	C1CC[C@H]([C@@H](C1)CN2CCN(CC2)C3=NSC4=CC=CC=C43)CN5C(=O)[C@H]6[C@@H]7CC[C@@H](C7)[C@H]6C5=O