产品详情
LY-2584702 hydrochloride is a selective ATP competitive inhibitor of p70S6K with an IC50 of 4 nM. In S6K1 enzyme assay, the IC50 of LY-2584702 is 2 nM.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 20.75 mL | 103.76 mL | 207.52 mL |
0.5 mM | 4.15 mL | 20.75 mL | 41.5 mL |
1 mM | 2.08 mL | 10.38 mL | 20.75 mL |
5 mM | 0.42 mL | 2.08 mL | 4.15 mL |
*The above data is based on the productmolecular weight 481.88. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
目录号 | A21416 |
---|---|
作用机制 | Inhibitor (抑制剂) |
M. Wt | 481.88 |
Formula | C21H20ClF4N7 |
Purity | >99% |
Storage | Store lyophilized at -20ºC, keep desiccated. |
CAS No. | 1082948-81-9 |
Synonyms | LY2584702, LY 2584702 |
SMILES | CN1C=C(C2=CC=C(F)C(C(F)(F)F)=C2)N=C1C3CCN(C4=C5C(NN=C5)=NC=N4)CC3.[H]Cl |
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