LY 379268
目录号: A13123
mGlu2 receptor 激动剂
LY 379268 是一种高度选择性的 group II mGlu 受体激动剂(对于 hmGlu2 和 hmGlu3 的 EC50 值分别为 2.69 和 4.48 nM),对 group I 和 group III 受体的选择性超过 80 倍。
Discription | LY 379268 is a highly selective group II mGlu receptor agonist (EC50 values are 2.69 and 4.48 nM for hmGlu2 and hmGlu3 respectively) that displays > 80-fold selectivity over group I and group III receptors. |
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目录号 | A13123 |
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分子式 | C7H9NO5 |
分子量 | 187.15 |
CAS号 | 191471-52-0 |
SMILES | C1[C@]([C@@H]2[C@H]([C@@H]2O1)C(=O)O)(C(=O)O)N |
其他名称 | LY379268, LY-379268 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2