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TGF-??R 抑制剂

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产品目录号: A11017


产品名 目录号 价格 数量
LY2157299 5mg A11017-5
¥ 900.00
LY2157299 10mg A11017-10
¥ 1,350.00
LY2157299 25mg A11017-25
¥ 2,700.00
LY2157299 100mg A11017-100
¥ 7,500.00
LY2157299 10mM * 1mL in DMSO A11017-10mM-D
¥ 1,250.00



LY2157299 is an orally active transforming growth factor beta receptor (TGF-βR) kinase inhibitor.





顾客使用 Adooq 产品发表的高质量科研文献
Adooq 顾客使用 LY2157299 发表的文献 (1)
  • Oguri G, .et al. Effects of methylglyoxal on human cardiac fibroblast: roles of transient receptor potential ankyrin 1 (TRPA1) channels., Am J Physiol Heart Circ Physiol., 2014, 307(9):H1339-52 PMID: 25172898

Chemical Information

目录号 A11017
Mechanism of action Inhibitor
分子量 369.4
化学分子式 C22H19N5O
Solubility DMSO
纯度 >98%
储存方式 at -20°C 2 years
CAS No. 700874-72-2
Synonyms LY-2157299
化学名称 4-[5,6-Dihydro-2-(6-methyl-2-pyridinyl)-4H-pyrrolo[1,2-b]pyrazol-3-yl]-6-quinolinecarboxamide


LY2157299 is an orally active transforming growth factor beta receptor (TGF-βR) kinase inhibitor.
TβRI (Cell-free assay)
56 nM


Solubility (25°C)* In vitro DMSO 74 mg/mL (200.31 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.


Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 27.07 mL 135.35 mL 270.71mL
0.5 mM 5.41 mL 27.07 mL 54.14 mL
1 mM 2.71 mL 13.54 mL 27.07 mL
5 mM 0.54 mL 2.71 mL 5.41 mL

*The above data is based on the productmolecular weight 369.4. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

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