LY2365109 hydrochloride
目录号: A21779
GlyT1 抑制剂
LY2365109 hydrochloride 是一种强效且选择性的 GlyT1 抑制剂,在过表达 hGlyT1a 的细胞中抑制甘氨酸摄取的 IC50 为 15.8 nM。
Discription | LY2365109 hydrochloride is a potent and selective GlyT1 inhibitor, with an IC50 of 15.8 nM for glycine uptake in cells over-expressing hGlyT1a. | ||
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目录号 | A21779 |
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分子式 | C22H28ClNO5 |
分子量 | 421.91 |
CAS号 | 1779796-27-8 |
SMILES | O=C(O)CN(CCOC1=CC=C(C2=CC=C(OCO3)C3=C2)C=C1C(C)(C)C)C.Cl[H] |
其他名称 | LY-2365109, LY 2365109 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2