LY317615 (Enzastaurin)

目录号: A10356

PKCβ inhibitor

LY317615 (Enzastaurin)

LY317615 (Enzastaurin) Chemical Structure

CAS NO. 170364-57-5

LY317615 (Enzastaurin) is a potent and selective inhibitor of PKCβ with antiproliferative activity (IC50= ~6 nM).

库存: 现货

规格 价格 数量
10 mg
¥ 400.00
50 mg
¥ 1,200.00
100 mg
¥ 2,000.00
200 mg
¥ 3,500.00
10mM * 1mL in DMSO
¥ 800.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

详情

LY317615 (Enzastaurin) is a potent and selective inhibitor of PKCβ with antiproliferative activity (IC50= ~6 nM).
Targets
PKCβ (Cell-free assay) PKCα (Cell-free assay) PKCγ (Cell-free assay) PKCε (Cell-free assay)
6 nM39 nM83 nM110 nM
In vitro (25°C) DMSO 30 mg/mL (58.18 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 15% Captisol 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 19.39 mL 96.97 mL 193.95 mL
0.5 mM 3.88 mL 19.39 mL 38.79 mL
1 mM 1.94 mL 9.7 mL 19.39 mL
5 mM 0.39 mL 1.94 mL 3.88 mL

*The above data is based on the productmolecular weight 515.6 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A10356
MECHANISM OF ACTION Inhibitor
M. Wt 515.6
Formula C32H29N5O2
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 170364-57-5
Synonyms LY-317615
SMILES CN1C=C(C2=CC=CC=C21)C3=C(C(=O)NC3=O)C4=CN(C5=CC=CC=C54)C6CCN(CC6)CC7=CC=CC=N7

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