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LY317615 (Enzastaurin)

促销

PKC?? 抑制剂

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产品目录号: A10356

库存状态:中国现货中国现货

产品名 目录号 价格 数量
LY317615 10mg A10356-10
¥ 400.00
LY317615 50mg A10356-50
¥ 1,200.00
LY317615 100mg A10356-100
¥ 2,000.00
LY317615 200mg A10356-200
¥ 3,500.00
LY317615 (Enzastaurin) 10mM * 1mL in DMSO A10356-10mM-D
¥ 800.00

产品仅用于研究,不针对患者销售,望谅解.

产品简介

LY317615 (Enzastaurin) is a potent and selective inhibitor of PKCβ with antiproliferative activity (IC50= ~6 nM).

LY317615 (Enzastaurin)

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Chemical Information

目录号 A10356
Mechanism of action Inhibitor
分子量 515.6
化学分子式 C32H29N5O2
Solubility DMSO
纯度 >98%
储存方式 at -20°C 2 years
CAS No. 170364-57-5
Synonyms LY-317615
SMILES code CN1C=C(C2=CC=CC=C21)C3=C(C(=O)NC3=O)C4=CN(C5=CC=CC=C54)C6CCN(CC6)CC7=CC=CC=N7
化学名称 3-(1-Methylindol-3-yl)-4-[1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]indol-3-yl]pyrrole-2,5-dione

生物活性

Description
LY317615 (Enzastaurin) is a potent and selective inhibitor of PKCβ with antiproliferative activity (IC50= ~6 nM).
Targets
PKCβ (Cell-free assay) PKCα (Cell-free assay) PKCγ (Cell-free assay) PKCε (Cell-free assay)
6 nM39 nM83 nM110 nM

溶解性

Solubility (25°C) * In vitro DMSO 30 mg/mL (58.18 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 15% Captisol 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 19.39 mL 96.97 mL 193.95mL
0.5 mM 3.88 mL 19.39 mL 38.79 mL
1 mM 1.94 mL 9.7 mL 19.39 mL
5 mM 0.39 mL 1.94 mL 3.88 mL

*The above data is based on the productmolecular weight 515.6 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

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