Lys-Des-Arg9Bradykinin
目录号: A23518
bradykinin B1 receptor 激动剂
Lys-[Des-Arg9]Bradykinin,一种天然存在的激肽,是一种高效且高度选择性的布拉迪肯B1受体激动剂,其Ki值分别为人类、小鼠和兔子B1受体的0.12 nM、1.7 nM和0.23 nM。Lys-[Des-Arg9]Bradykinin对B2受体的抑制活性较低。
bradykinin B1 receptor 激动剂
Discription | Lys-[Des-Arg9]Bradykinin, a naturally occurring kinin, is a potent and highly selective bradykinin B1 receptor agonist with a Ki of 0.12 nM, 1.7 nM and 0.23 nM for human, mouse and rabbit B1 receptors, respectively. Lys-[Des-Arg9]Bradykinin has low inhibitory activity on B2 receptors. | |||||
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Cell Research |
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目录号 | A23518 |
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分子式 | C50H73N13O11 |
分子量 | 1032.2 |
CAS号 | 71800-36-7 |
Sequence | Lys-Arg-Pro-Pro-Gly-Phe-Ser-Pro-Phe |
Sequence shortening | KRPPGFSPF |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2