Mardepodect
目录号: A20641
PDE10A 抑制剂
Mardepodect(PF-2545920)是一种强效的、口服活性的、选择性的 PDE10A 抑制剂,其 IC50 为 0.37 nM,对其他 PDEs 的选择性超过1000倍。Mardepodect 能够穿越血脑屏障。
Discription | Mardepodect (PF-2545920) is a potent, orally active and selective PDE10A inhibitor with an IC50 of 0.37 nM, with >1000-fold selectivity over other PDEs. Mardepodect can cross the blood-brain barrier. | |||||
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Cell Research |
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目录号 | A20641 |
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分子式 | C25H20N4O |
分子量 | 392.45 |
CAS号 | 898562-94-2 |
SMILES | CN(N=C1C2=CC=C(OCC3=NC4=CC=CC=C4C=C3)C=C2)C=C1C5=CC=NC=C5 |
其他名称 | PF-2545920, PF2545920, PF 2545920 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2