Mavatrep
目录号: A15778
TRPV1 拮抗剂
Mavatrep 是一种口服生物利用度的 TRPV1 拮抗剂(Ki=6.5 nM),对 CYP 同工酶 3A4、1A2 和 2D6 的酶活性几乎没有影响(IC50 > 25 μM)。
Discription | Mavatrep is an orally bioavailable TRPV1 antagonist (Ki=6.5 nM), exhibits minimal effect on the enzymatic activity (IC50 > 25 μM) of CYP isoforms 3A4, 1A2, and 2D6. | |||||
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Cell Research |
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目录号 | A15778 |
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分子式 | C25H21F3N2O |
分子量 | 422.44 |
CAS号 | 956274-94-5 |
SMILES | CC(C)(C1=CC=CC=C1C2=CC3=C(C=C2)N=C(N3)C=CC4=CC=C(C=C4)C(F)(F)F)O |
其他名称 | JNJ-39439335 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2