Miransertib hydrochloride
目录号: A22376
Akt 抑制剂
Miransertib hydrochloride (ARQ-092 hydrochloride) 是一种强效的、口服活性的、选择性的和烷基Akt抑制剂,其IC50分别为Akt1的2.7 nM、Akt2的14 nM和Akt3的8.1 nM。
Discription | Miransertib hydrochloride (ARQ-092 hydrochloride) is a potent, orally active, selective and allosteric Akt inhibitor with IC50s of 2.7 nM, 14 nM and 8.1 nM for Akt1, Akt2, Akt3, respectively. | |||||
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Cell Research |
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目录号 | A22376 |
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分子式 | C27H25ClN6 |
分子量 | 468.98 |
CAS号 | 1313883-00-9 |
SMILES | NC1=NC=CC=C1C2=NC3=CC=C(C4=CC=CC=C4)N=C3N2C5=CC=C(C6(N)CCC6)C=C5.[H]Cl |
其他名称 | ARQ-092 hydrochloride, ARQ092, ARQ 092 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2