Mozavaptan

Name: Mozavaptan
SKU: A16622

目录号: A16622

nonpeptide vasopressin V2 receptor antagonist

Mozavaptan Chemical Structure

CAS NO. 137975-06-5

Mozavaptan (OPC31260) is a orally effective, nonpeptide vasopressin V2 receptor antagonist with an IC50 of 14 nM.

库存：现货

规格	价格	数量
10 mg	￥ 540.00
25 mg	￥ 1,080.00
50 mg	￥ 1,860.00
100 mg	￥ 3,180.00

大包装询价

或

添加到收藏

产品仅用于科学研究，不针对患者销售，望谅解.

产品详情

生物活性

Mozavaptan (OPC31260) is a orally effective, nonpeptide vasopressin V2 receptor antagonist with an IC50 of 14 nM.

溶解度 *

In vitro (25°C)	DMSO	1 mg/mL (2.33 mM)
	Water	Insoluble
	Ethanol	1 mg/mL (2.33 mM)
In vivo	30% propylene glycol, 5% Tween 80, 65% D5W	28 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	23.39 mL	116.95 mL	233.9 mL
0.5 mM	4.68 mL	23.39 mL	46.78 mL
1 mM	2.34 mL	11.69 mL	23.39 mL
5 mM	0.47 mL	2.34 mL	4.68 mL

*The above data is based on the productmolecular weight 427.54. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A16622
作用机制	Antagonist (拮抗剂)
M. Wt	427.54
Formula	C27H29N3O2
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	137975-06-5
SMILES	CC1=CC=CC=C1C(NC2=CC=C(C(N3C(C=CC=C4)=C4C(N(C)C)CCC3)=O)C=C2)=O